Synthesis of Arylated Quinolines by Chemo- and Site-selective Suzuki–Miyaura Reactions of 5,7-Dibromo-8-(trifluoromethanesulfonyloxy)Quinoline

Eleya, Nadi and Mahal, Ahmed and Hein, Martin and Villinger, Alexander and Langer, Peter (2011) Synthesis of Arylated Quinolines by Chemo- and Site-selective Suzuki–Miyaura Reactions of 5,7-Dibromo-8-(trifluoromethanesulfonyloxy)Quinoline. Advanced Synthesis & Catalysis, 353 (14-15). pp. 2761-2774. ISSN 1615-4169 (online)

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Abstract

Arylated quinolines were prepared by Suzuki–Miyaura reactions of 5,7-dibromo-8-(trifluoromethanesulfonyloxy)quinoline. The reactions proceed with excellent site-selectivity. The first, second and third attack occur at positions 5, 7 and 8, respectively.

Item Type: Article
Uncontrolled Keywords: Arylated quinolines; Suzuki–Miyaura reaction; Site-selective cross-coupling
Subjects: Q Science > QD Chemistry
T Technology > TP Chemical technology
Divisions: Department of Medical Biochemical Analysis > Research papers
Depositing User: ePrints Depositor
Date Deposited: 13 Aug 2025 11:19
Last Modified: 13 Aug 2025 11:19
URI: https://eprints.cihanuniversity.edu.iq/id/eprint/4742

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